SCHEMBL8307936

SCHEMBL8307936

CN(CCOc1ccc(Cl)c2c1CC(=O)N2)c1cccs1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.39
PDE4D Q08499 2/20 0.39
PDE7A Q13946 2/20 0.39
PDE1A P54750 1/20 0.39
PDE1B Q01064 1/20 0.39
PDE1C Q14123 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310167 0.81 PDE5A (0.39) PDE5APDE4DPDE7APDE1APDE1B
SCHEMBL7470775 0.76 ATM (0.49)
SCHEMBL7458470 0.74 DRD2 (0.48)
SCHEMBL7207588 0.73 SLC6A9 (0.32)
SCHEMBL7470200 0.68 POLB (0.45)
SCHEMBL7475432 0.67 DRD2 (0.68)
SCHEMBL7457321 0.66 DRD2 (0.49)
SCHEMBL7478885 0.65 DRD2 (0.54)
SCHEMBL14507273 0.65
SCHEMBL7476726 0.65 DRD2 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923576-A1 4-AMINOETHOXY-INDOLONE DERIVATIVES AS DOPAMINE D2 AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-06-23 EP claimed
WO-1998008843-A1 4-AMINOETHOXY-INDOLONE DERIVATIVES AS DOPAMINE D2 AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 1998-03-05 WO claimed