SCHEMBL8307946

SCHEMBL8307946

Cc1nc(-c2nc(-c3ccc(Cl)cc3)c(CCO)o2)c[nH]1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
AKT1 P31749 1/20 0.33
TARBP2 Q15633 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
NOTUM Q6P988 1/20 0.32
CRHR1 P34998 1/20 0.32
RXRA P19793 3/20 0.31
RXRB P28702 3/20 0.31
RXRG P48443 3/20 0.31
PTGS2 P35354 1/20 0.31
KDM4E B2RXH2 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
LMNA P02545 1/20 0.31
PDGFRB P09619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4442406 0.93 SIRT2 (0.38) ALDH1A1NPSR1AKT1TARBP2SIRT2
SCHEMBL4563793 0.92 SIRT2 (0.35) ALDH1A1NPSR1AKT1TARBP2SIRT2
SCHEMBL4442084 0.91 SIRT2 (0.34) ALDH1A1NPSR1AKT1TARBP2SIRT2
SCHEMBL7514117 0.91 SIRT2 (0.34) ALDH1A1NPSR1AKT1TARBP2SIRT2
SCHEMBL8305905 0.86 RXRA (0.45) ALDH1A1RXRARXRBRXRGKDM4E
SCHEMBL8303146 0.86 CRHR1 (0.31) CRHR1
SCHEMBL8303347 0.85 NR4A2 (0.35) ALDH1A1TARBP2RXRARXRBRXRG
SCHEMBL8303834 0.85 CYP1A2 (0.32) ALDH1A1NPSR1CRHR1PTGS2KDM4E
SCHEMBL8303845 0.85 RXRA (0.41) ALDH1A1RXRARXRBRXRGPTGS2
SCHEMBL7510444 0.81 PTGS1 (0.34) NOTUMRXRARXRBRXRGPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891340-A1 OXAZOLE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1999-01-20 EP disclosed
WO-1997036882-A1 OXAZOLE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-09 WO disclosed