SCHEMBL8553140

SCHEMBL8553140

Nc1ccc2oc(C(=O)c3ccncc3)c(CCC(=O)O)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 8/20 0.39
NPC1 O15118 7/20 0.39
RAB9A P51151 6/20 0.39
SMN1; SMN2 Q16637 6/20 0.39
CASP1 P29466 2/20 0.39
ADORA2A P29274 1/20 0.39
KDM4E B2RXH2 7/20 0.39
ALDH1A1 P00352 7/20 0.39
HPGD P15428 5/20 0.39
HSD17B10 Q99714 4/20 0.39
KMT2A Q03164 3/20 0.39
GFER P55789 1/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2C9 P11712 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
TDP1 Q9NUW8 3/20 0.36
MEN1 O00255 2/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553130 0.91 ALDH1A1 (0.38) MAPTNPC1RAB9ASMN1; SMN2CASP1
SCHEMBL8308345 0.86 ALDH1A1 (0.49) MAPTNPC1RAB9ASMN1; SMN2CASP1
SCHEMBL8305025 0.81 ALDH1A1 (0.41) MAPTNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL8837860 0.80 KDM4E (0.52) CASP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8308344 0.77 ALDH1A1 (0.47) MAPTNPC1RAB9ASMN1; SMN2CASP1
SCHEMBL8305023 0.75 ALDH1A1 (0.44) MAPTRAB9ASMN1; SMN2CASP1KDM4E
SCHEMBL16547892 0.73 MAPT (0.57) MAPTNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL10556380 0.69 CYP2C9 (0.58) MAPTNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL8307015 0.68 KDM4E (0.46) MAPTNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL8307605 0.68 MAPK1 (0.39) MAPTCASP1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685474-B1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1998-09-16 EP disclosed
US-5565488-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US disclosed
EP-0685474-A1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed