SCHEMBL8553130

SCHEMBL8553130

Nc1ccc2c(CCC(=O)O)c(C(=O)c3ccncc3)oc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.38
KDM4E B2RXH2 6/20 0.38
HPGD P15428 5/20 0.38
HSD17B10 Q99714 3/20 0.38
CASP1 P29466 2/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 1/20 0.38
CASP7 P55210 1/20 0.38
MAPT P10636 6/20 0.36
TDP1 Q9NUW8 2/20 0.36
NPC1 O15118 3/20 0.36
KMT2A Q03164 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP2C9 P11712 2/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
NPSR1 Q6W5P4 3/20 0.35
ALOX12 P18054 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553140 0.91 MAPT (0.39) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL8837860 0.87 KDM4E (0.52) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL8308344 0.86 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL8305023 0.81 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL8307605 0.77 MAPK1 (0.39) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL8308345 0.77 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL8305025 0.75 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDHSD17B10GAA
SCHEMBL8837925 0.74 KDM4E (0.48) ALDH1A1KDM4EHPGDHSD17B10CASP1
SCHEMBL27445439 0.73 SMN1; SMN2 (0.43) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL16547892 0.73 MAPT (0.57) ALDH1A1KDM4EHPGDTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0685474-B1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1998-09-16 EP disclosed
US-5565488-A ANTIINFLAMMATORY AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1996-10-15 US disclosed
EP-0685474-A1 Oxalylamino-benzofuran- and benzothienyl-derivatives BAYER AG (DE) 1995-12-06 EP disclosed