SCHEMBL8308620

SCHEMBL8308620

CS(=O)(=O)c1ccc(-c2cc3cc(-c4ccccc4F)ccc3[nH]2)cc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCD O00767 5/20 0.55
FADS1 O60427 1/20 0.55
CDK5 Q00535 2/20 0.49
CDK5R1 Q15078 2/20 0.49
PTGS2 P35354 5/20 0.49
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA9 Q16790 2/20 0.48
PRKDC P78527 1/20 0.47
ATM Q13315 1/20 0.47
ATR Q13535 1/20 0.47
TRPA1 O75762 1/20 0.45
FFAR1 O14842 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8444391 0.81 CDK5 (0.55) CDK5CDK5R1PTGS2CA12CA1
SCHEMBL8306238 0.81 CDK5 (0.60) SCDCDK5CDK5R1PTGS2CA12
SCHEMBL8305443 0.80 CA12 (0.72) CDK5CDK5R1PTGS2CA12CA1
SCHEMBL9206986 0.78 PTGS2 (0.73) SCDFADS1PTGS2
SCHEMBL8306286 0.77 CDK5 (0.56) CDK5CDK5R1PTGS2CA12CA1
SCHEMBL8308055 0.76 MEN1 (0.60) CDK5CDK5R1PTGS2CA12CA1
SCHEMBL1460085 0.75 KIF11 (0.42) SCDFADS1CDK5CDK5R1PTGS2
SCHEMBL8307211 0.75 CA12 (0.57) PTGS2CA12CA1CA2CA9
SCHEMBL4154662 0.73 FFAR1 (0.54) SCDFADS1CA12CA1CA2
SCHEMBL8522642 0.72 PTGS2 (0.63) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915848-A1 1,2-DIARYLINDOLE AS COX-2 INHIBITORS LABORATOIRES UPSA (FR) 1999-05-19 EP claimed
WO-1998005639-A1 1,2-DIARYLINDOLE AS COX-2 INHIBITORS LABORATOIRES UPSA (FR) 1998-02-12 WO claimed