SCHEMBL8309915

SCHEMBL8309915

O=c1c(Br)ccccc1N1CCNCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.56
ADRB1 P08588 3/20 0.55
HTR1A P08908 4/20 0.50
HTR7 P34969 3/20 0.50
HTR3A P46098 3/20 0.50
HTR2A P28223 2/20 0.50
HTR5A P47898 2/20 0.50
HTR3E A5X5Y0 2/20 0.50
HTR3B O95264 2/20 0.50
HTR3D Q70Z44 2/20 0.50
HTR3C Q8WXA8 2/20 0.50
SIGMAR1 Q99720 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
NCF1 P14598 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
HTR1D P28221 1/20 0.50
HTR1B P28222 1/20 0.50
MTOR P42345 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL8313245 0.91 HTR6 (0.55) HTR6ADRB1HTR1AHTR7HTR3A
SCHEMBL29446041 0.89 HTR6 (0.62) HTR6ADRB1HTR1AHTR7HTR3A
SCHEMBL10677139 0.89 HTR6 (0.62) HTR6ADRB1HTR1AHTR7HTR3A
SCHEMBL232830 0.89 HTR6 (0.62) HTR6ADRB1HTR1AHTR7HTR3A
Hydrochloric Acid SCHEMBL27845681 0.87 HTR6 (0.61) HTR6ADRB1HTR1AHTR7HTR3A
Piperazine SCHEMBL28234322 0.87 HTR6 (0.61) HTR6ADRB1HTR1AHTR7HTR3A
Ethane SCHEMBL11509421 0.85 ADRB1 (0.61) HTR6ADRB1HTR1AHTR7HTR3A
SCHEMBL11087855 0.79 ADRA2C (0.53) HTR6HTR1AHTR2ANCF1TSHR
SCHEMBL15834279 0.78 ADRB1 (0.75) HTR6ADRB1HTR1AHTR7HTR3A
SCHEMBL7582175 0.78 HTR6 (0.54) HTR6ADRB1HTR1AHTR7HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998414-A PSYCHOLOGICAL DISORDERS HOECHST MARION ROUSSEL, INC. (US) 1999-12-07 US disclosed
EP-0929537-A1 TROPONYL PIPERAZINES AS SELECTIVE DOPAMINE D4 RECEPTOR LIGANDS HOECHST MARION ROUSSEL, INC. (US) 1999-07-21 EP disclosed
WO-1998007711-A1 TROPONYL PIPERAZINES AS SELECTIVE DOPAMINE D4 RECEPTOR LIGANDS HOECHST MARION ROUSSEL, INC. (US) 1998-02-26 WO disclosed