SCHEMBL8310773

SCHEMBL8310773

CC(C)C(=O)C(=O)c1cccs1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.72
CES1 P23141 2/20 0.72
RAB9A P51151 6/20 0.55
ALDH1A1 P00352 5/20 0.55
NPC1 O15118 5/20 0.55
HPGD P15428 3/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
DAO P14920 1/20 0.52
KMT2A Q03164 3/20 0.48
LMNA P02545 2/20 0.48
MEN1 O00255 2/20 0.48
POLB P06746 1/20 0.48
HDAC1 Q13547 1/20 0.48
CYP2C9 P11712 2/20 0.46
KDM4E B2RXH2 1/20 0.46
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
KEAP1 Q14145 1/20 0.46
HPGDS O60760 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1066873 0.85 CES2 (1.00) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL6417954 0.82 CES2 (0.57) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL19388239 0.82 CES2 (0.57) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL7640314 0.79 CES2 (0.59) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL619898 0.79 CES2 (0.64) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL2610951 0.77 CES2 (0.74) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL6415141 0.77 CES2 (0.55) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL14782239 0.77 CES2 (0.55) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL9148741 0.76 CES2 (0.81) CES2CES1RAB9AALDH1A1NPC1
SCHEMBL1937375 0.75 RAB9A (0.58) CES2CES1RAB9AALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9770439-B2 Hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2017-09-26 US disclosed
US-9770439-B2 Hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2017-09-26 US disclosed
US-20160199355-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL MAYERS SQUIBB COMPANY (US) 2016-07-14 US disclosed
US-20160158200-A1 Combinations of Hepatitis C Virus Inhibitors BRISTOL MYERS SQUIBB CO (US) 2016-06-09 US disclosed
US-9326973-B2 Hepatitis C virus inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2016-05-03 US disclosed
US-20150297568-A1 Hepatitis C Virus Inhibitors BRISTOL MYERS SQUIBB CO (US) 2015-10-22 US disclosed
US-20150023913-A1 Hepatitis C Virus Inhibitors BRISTOL-MYERS SQUIBB COMPANY 2015-01-22 US disclosed
US-20130183269-A1 Hepatitis C Virus Inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2013-07-18 US disclosed
US-7217794-B2 Compounds and methods for treatment of thrombosis DAIAMED, INC. (US) 2007-05-15 US disclosed
WO-2004089297-A2 COMPOUNDS AND METHODS FOR TREATMENT OF THROMBOSIS SUNTORY PHARMACEUTICAL RESEARCH LABORATORIES, LLC (US) 2004-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130183269-A1 Hepatitis C Virus Inhibitors HAVCR2, MAVS, EIF2AK2 CES2 1947/4885CES1 536/4885RAB9A 1490/4885
US-20160199355-A1 HEPATITIS C VIRUS INHIBITORS HAVCR2, MAVS, EIF2AK2 CES2 1947/4885CES1 536/4885RAB9A 1490/4885
US-20150023913-A1 Hepatitis C Virus Inhibitors HAVCR2, MAVS, EIF2AK2 CES2 1947/4885CES1 536/4885RAB9A 1490/4885
US-20150297568-A1 Hepatitis C Virus Inhibitors HAVCR2, MAVS, EIF2AK2 CES2 1947/4885CES1 536/4885RAB9A 1490/4885
US-20160158200-A1 Combinations of Hepatitis C Virus Inhibitors HAVCR2, EIF2AK2, MAVS CES2 1832/4885CES1 685/4885RAB9A 1807/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.