SCHEMBL8310871

SCHEMBL8310871

CC1(C)C=C(c2cccc[n+]2[O-])c2cc(S(C)(=O)=O)ccc2OC1

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 2/20 0.40
ABCC8 Q09428 2/20 0.40
KCNJ11 Q14654 2/20 0.40
KCNJ8 Q15842 2/20 0.40
PKM P14618 1/20 0.34
DAO P14920 1/20 0.32
PTGS2 P35354 5/20 0.32
PTGS1 P23219 2/20 0.32
MGAT2 Q10469 1/20 0.32
MAP3K5 Q99683 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310333 0.89 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8PKM
SCHEMBL8310464 0.84 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8314327 0.84 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8312815 0.83 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8310409 0.83 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8MGAT2
SCHEMBL8316384 0.82 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8311451 0.82 HTR2B (0.39) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8315805 0.81 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8313863 0.81 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8315406 0.81 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP claimed
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5652252-A POTASSIUM CHANNEL ACTIVATORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-07-29 US disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
EP-0626954-A1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GmbH (DE) 1994-12-07 EP disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed