SCHEMBL8310333

SCHEMBL8310333

CC1(C)C=C(c2cccc[n+]2[O-])c2cc(S(=O)(=O)c3ccccc3)ccc2OC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 2/20 0.39
ABCC8 Q09428 2/20 0.39
KCNJ11 Q14654 2/20 0.39
KCNJ8 Q15842 2/20 0.39
HTR6 P50406 5/20 0.38
PKM P14618 1/20 0.33
ABCB1 P08183 3/20 0.32
ABCC1 P33527 3/20 0.32
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
MGAT2 Q10469 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
NLRP3 Q96P20 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310871 0.89 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8PKM
SCHEMBL8311451 0.82 HTR2B (0.39) ABCC9ABCC8KCNJ11KCNJ8HTR2B
SCHEMBL8310464 0.82 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8MAPT
SCHEMBL8314327 0.82 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8HTR2C
SCHEMBL8313863 0.81 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8ALDH1A1
SCHEMBL8310409 0.81 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8HTR6
SCHEMBL8312815 0.81 ABCC9 (0.39) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8316384 0.80 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8315805 0.79 ABCC9 (0.38) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8314966 0.79 KDM4E (0.39) ABCC9ABCC8KCNJ11KCNJ8ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP claimed
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5652252-A POTASSIUM CHANNEL ACTIVATORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-07-29 US disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
EP-0626954-A1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GmbH (DE) 1994-12-07 EP disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed