SCHEMBL8311679

SCHEMBL8311679

CC(N)(C(=O)O)c1csc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.45
MAPT P10636 2/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
ALOX5 P09917 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CYP2A6 P11509 3/20 0.41
CNR2 P34972 1/20 0.40
PTPN7 P35236 1/20 0.38
DUSP3 P51452 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313877 0.85 PKM (0.46) PKMMAPTHDAC3HDAC4HDAC1
SCHEMBL3191250 0.85 PKM (0.46) PKMMAPTHDAC3HDAC4HDAC1
SCHEMBL8313331 0.79 PIN1 (0.39) PKMMAPTHDAC3HDAC4HDAC1
SCHEMBL6671866 0.79 PKM (0.44) PKMMAPTHDAC3HDAC4HDAC1
Hydrochloric Acid SCHEMBL8312738 0.78 PIN1 (0.38) PKMMAPTHDAC3HDAC4HDAC1
SCHEMBL74015 0.76 MAPT (0.48) PKMMAPTHDAC3HDAC4HDAC1
SCHEMBL9764850 0.75 ALOX5 (0.51) PKMMAPTHDAC3HDAC4HDAC1
SCHEMBL6844569 0.75 CYP2A6 (0.49) PKMMAPTHDAC3HDAC4HDAC1
SCHEMBL4232293 0.74 PKM (0.46) PKMMAPTHDAC3HDAC4HDAC1
SCHEMBL10559844 0.74 ALOX5 (0.50) PKMMAPTHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635508-B1 TETRAHYDROPYRIDINE DERIVATIVE HAVING SUBSTITUENTS ON THREE RINGS ASAHI CHEMICAL IND (JP) 1999-10-06 EP disclosed
US-5621103-A 3-(SUBSTITUTED METHYLAMINOCARBONYL)-1,2,3,4-TETRAHYDRO-(1)BENZOTHIENO(2,3-C) PYRIDINES; ANXIOLYTIC AGENTS; LEARNING ENHANCEMENT ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1997-04-15 US disclosed
EP-0635508-A1 TETRAHYDROPYRIDINE DERIVATIVE HAVING SUBSTITUENTS ON THREE RINGS Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1995-01-25 EP disclosed
EP-0386258-A1 TETRAHYDROPYRIDINE DERIVATIVES Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1990-09-12 EP disclosed