SCHEMBL8312333

SCHEMBL8312333

Cc1cc2c(=O)[nH][nH]c(=O)c2n1CC(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.39
TSHR P16473 2/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
ALDH1A1 P00352 6/20 0.36
ADRA2A P08913 1/20 0.36
DAO P14920 2/20 0.35
KDM4E B2RXH2 5/20 0.34
MAPT P10636 2/20 0.34
THRB P10828 1/20 0.34
TP53 P04637 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
B3GNT2 Q9NY97 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4763472 0.69 ALDH1A1 (0.47) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1
SCHEMBL8315752 0.69 MEN1 (0.39) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1
SCHEMBL29776965 0.67 B3GNT2 (0.43) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1
SCHEMBL6394776 0.67 ALDH1A1 (0.67) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1
SCHEMBL8317250 0.67 ALDH1A1 (0.32) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1
SCHEMBL9739218 0.63 ALDH1A1 (0.43) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1
SCHEMBL11637797 0.60 KDM4E (0.77) HSD17B10KMT2AMEN1ALDH1A1KDM4E
SCHEMBL4767676 0.60 B3GNT2 (0.43) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1
SCHEMBL11429505 0.59 RGS4 (0.50) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1
SCHEMBL20853011 0.59 CCR2 (0.38) SMN1; SMN2TSHRHSD17B10TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609328-B1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-28 EP disclosed
US-5534515-A Pyrrolopyridazines having gastrointestinal protective effects BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-07-09 US disclosed
WO-1993008190-A1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1993-04-29 WO disclosed