SCHEMBL8312860

SCHEMBL8312860

CCc1ccc(-c2nc3ccc(S(=O)(=O)C4(C(=O)NOC5CCCCO5)CCOCC4)cc3s2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.37
KDM4E B2RXH2 4/20 0.36
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
NPC1 O15118 3/20 0.36
HPGD P15428 3/20 0.36
RAB9A P51151 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
ALDH1A1 P00352 4/20 0.36
MMP13 P45452 5/20 0.36
MMP1 P03956 3/20 0.36
MMP9 P14780 3/20 0.36
ADAM17 P78536 1/20 0.36
HDAC6 Q9UBN7 1/20 0.35
MMP2 P08253 4/20 0.35
MMP8 P22894 4/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6267605 0.94 MMP13 (0.37) RORCKDM4EKMT2AMEN1NPC1
SCHEMBL6230548 0.93 MMP13 (0.41) RORCKDM4EKMT2AMEN1NPC1
SCHEMBL8312513 0.92 MMP13 (0.45) RORCMMP13MMP1MMP9ADAM17
SCHEMBL6278357 0.91 MMP8 (0.46) RORCMMP13MMP1MMP9MMP2
SCHEMBL6234746 0.90 MMP2 (0.44) RORCKMT2AALDH1A1MMP13MMP1
SCHEMBL6276528 0.89 ALDH1A1 (0.37) RORCKMT2AMEN1NPC1HPGD
SCHEMBL6230523 0.88 MMP2 (0.46) RORCKDM4EKMT2ASMN1; SMN2ALDH1A1
SCHEMBL6231050 0.88 ALDH1A1 (0.34) KDM4EKMT2ASMN1; SMN2ALDH1A1MMP13
SCHEMBL6231944 0.88 ALDH1A1 (0.39) KDM4EKMT2AMEN1NPC1HPGD
SCHEMBL6229096 0.85 MMP2 (0.44) KMT2ASMN1; SMN2ALDH1A1MMP13MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004048368-A2 HETEROARYLSULFONYLMETHYL HYDROXAMIC ACIDS AND AMIDES AND THEIR USE AS PROTEASE INHIBITORS PHARMACIA CORPORATION (US) 2004-06-10 WO disclosed