SCHEMBL8315996

SCHEMBL8315996

CC1(C)COc2cc(Cl)c(F)cc2C(O)(c2ccccn2)C1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.35
SCN9A Q15858 3/20 0.34
OPRM1 P35372 1/20 0.34
AKR1B1 P15121 1/20 0.33
BACE1 P56817 3/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
NR3C1 P04150 1/20 0.32
GRM4 Q14833 1/20 0.31
ADAMTS4 O75173 1/20 0.31
MMP2 P08253 1/20 0.31
MMP14 P50281 1/20 0.31
ADAM17 P78536 1/20 0.31
ADAMTS5 Q9UNA0 1/20 0.31
TRPV3 Q8NET8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316027 0.92 SCN9A (0.40) SLC6A2SCN9AOPRM1BACE1BACE2
SCHEMBL8313558 0.91 SLC6A2 (0.38) SLC6A2SCN9AOPRM1AKR1B1NR3C1
SCHEMBL8311266 0.85 SLC6A2 (0.37) SLC6A2AKR1B1BACE1TRPV3
SCHEMBL8313637 0.84 SLC6A2 (0.36) SLC6A2BACE1NR3C1
SCHEMBL8310494 0.81 SCN9A (0.38) SLC6A2SCN9A
SCHEMBL8311725 0.81 SLC6A2 (0.36) SLC6A2NR3C1
SCHEMBL8310708 0.81 SLC6A2 (0.40) SLC6A2OPRM1NR3C1
SCHEMBL8316835 0.81 SLC6A2 (0.39) SLC6A2OPRM1NR3C1
SCHEMBL8314947 0.80 SLC6A2 (0.37) SLC6A2SCN9A
SCHEMBL8314123 0.80 SLC6A2 (0.37) SLC6A2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed