SCHEMBL8313656

SCHEMBL8313656

Cc1cc2cn[nH]c(=O)c2n1Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.56
HSD17B10 Q99714 3/20 0.56
CYP1A2 P05177 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
TYMS P04818 5/20 0.55
TSHR P16473 4/20 0.52
ALDH1A1 P00352 3/20 0.52
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
USP2 O75604 1/20 0.49
LMNA P02545 2/20 0.48
MAPT P10636 1/20 0.48
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HPGD P15428 2/20 0.44
PSMD14 O00487 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312892 0.85 TYMS (0.58) KDM4ETYMSTSHRALDH1A1KMT2A
SCHEMBL8315752 0.76 MEN1 (0.39) KDM4EHSD17B10CYP1A2CYP2C9CYP2C19
SCHEMBL9740097 0.76 KDM4E (0.67) KDM4EHSD17B10CYP1A2CYP2C9CYP2C19
SCHEMBL8316752 0.72 TYMS (0.45) KDM4ECYP1A2CYP2C9CYP2C19TYMS
SCHEMBL15426106 0.72 KDM4E (1.00) KDM4EHSD17B10CYP1A2CYP2C9CYP2C19
SCHEMBL8313452 0.71 ALDH1A1 (0.56) KDM4EHSD17B10CYP1A2CYP2C9CYP2C19
SCHEMBL21407925 0.68 KDM4E (0.54) KDM4EHSD17B10CYP1A2CYP2C9CYP2C19
SCHEMBL13200852 0.68 HTR3A (0.61) KDM4EHSD17B10CYP1A2CYP2C9CYP2C19
SCHEMBL2475184 0.68 TYMS (0.46) KDM4ECYP1A2CYP2C9CYP2C19TYMS
SCHEMBL8318381 0.68 KMT2A (0.42) KDM4ECYP1A2CYP2C9CYP2C19L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609328-B1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEM FAB (DE) 1999-04-28 EP disclosed
US-5534515-A Pyrrolopyridazines having gastrointestinal protective effects BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-07-09 US disclosed
WO-1993008190-A1 PYRROLO-PYRIDAZINES WITH GASTRO-INTESTINAL PROTECTIVE ACTION BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1993-04-29 WO disclosed