SCHEMBL8314516

SCHEMBL8314516

CCCCOc1ccc(CN2CCC(N3CCC(C(=O)c4ccc(S(=O)(=O)c5ccc(O)c(O)c5)cc4)CC3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 9/20 0.52
CHRM1 P11229 6/20 0.51
CHRM3 P20309 2/20 0.51
CHRM4 P08173 1/20 0.51
S1PR5 Q9H228 3/20 0.50
HRH3 Q9Y5N1 4/20 0.46
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP2D6 P10635 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
SLC18A3 Q16572 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319668 0.97 CHRM2 (0.52) CHRM2CHRM1CHRM3CHRM4S1PR5
SCHEMBL8313975 0.92 CHRM2 (0.49) CHRM2CHRM1CHRM3CHRM4HRH3
SCHEMBL8314558 0.82 CHRM2 (0.55) CHRM2
SCHEMBL8314793 0.76 HRH3 (0.55) CHRM2HRH3MEN1ALDH1A1CYP2D6
SCHEMBL8313001 0.76 MEN1 (0.45) CHRM2S1PR5HRH3MEN1ALDH1A1
SCHEMBL8315643 0.75 CHRM2 (0.52) CHRM2
SCHEMBL8314512 0.75 CHRM2 (0.47) CHRM2CHRM1CHRM4S1PR5HRH3
SCHEMBL8315477 0.72 ALDH1A1 (0.51) CHRM2MEN1ALDH1A1KMT2A
SCHEMBL8791763 0.70 PRKAA2 (0.56) S1PR5HRH3MEN1ALDH1A1CYP2D6
SCHEMBL7409733 0.69 S1PR5 (0.63) S1PR5HRH3MEN1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004066960-A2 COMBINATION OF H1, H3 AND H4 RECEPTOR ANTAGONISTS FOR TREATMENT OF ALLERGIC AND NON-ALLERGIC PULMONARY INFLAMMATION, CONGESTION AND ALLERGIC RHINITIS SCHERING CORPORATION (US) 2004-08-12 WO disclosed