SCHEMBL8315477

SCHEMBL8315477

COc1ccc(CN2CCC(C3CCN(Cc4ccc(S(=O)(=O)c5ccc(O)c(O)c5)cc4)CC3)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
LMNA P02545 3/20 0.51
POLB P06746 2/20 0.51
MAPK1 P28482 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
KDM4E B2RXH2 2/20 0.48
NSD2 O96028 1/20 0.47
GAA P10253 1/20 0.47
GFER P55789 1/20 0.47
TSHR P16473 1/20 0.47
MMP1 P03956 1/20 0.47
MMP9 P14780 1/20 0.47
MMP13 P45452 1/20 0.47
ADAM17 P78536 1/20 0.47
CHRM2 P08172 1/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
ACHE P22303 1/20 0.45
SIGMAR1 Q99720 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314793 0.84 HRH3 (0.55) ALDH1A1CHRM2KMT2AMEN1
SCHEMBL8313001 0.84 MEN1 (0.45) ALDH1A1TSHRMMP1MMP9MMP13
SCHEMBL8314512 0.81 CHRM2 (0.47) ALDH1A1LMNAKDM4EMMP1MMP9
SCHEMBL7353607 0.79 S1PR5 (0.58) ALDH1A1LMNAPOLBMAPK1SMN1; SMN2
SCHEMBL9646910 0.79 PKM (0.68) POLBMAPK1NSD2GAAGFER
SCHEMBL8313087 0.78 CHRM2 (0.54) ALDH1A1LMNAPOLBGAACHRM2
SCHEMBL8313105 0.77 HDAC3 (0.52) KMT2AMEN1
SCHEMBL7347681 0.76 ALDH1A1 (0.64) ALDH1A1LMNAPOLBSMN1; SMN2KDM4E
SCHEMBL28213371 0.73 SIGMAR1 (0.55) ALDH1A1LMNAPOLBMAPK1SMN1; SMN2
Hydrochloric Acid SCHEMBL28859867 0.72 SIGMAR1 (0.54) ALDH1A1LMNAPOLBMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004066960-A2 COMBINATION OF H1, H3 AND H4 RECEPTOR ANTAGONISTS FOR TREATMENT OF ALLERGIC AND NON-ALLERGIC PULMONARY INFLAMMATION, CONGESTION AND ALLERGIC RHINITIS SCHERING CORPORATION (US) 2004-08-12 WO disclosed