SCHEMBL8315366

SCHEMBL8315366

O=CNCC(CCCN1C(=O)c2ccccc2C1=O)(c1ccccc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAOB P27338 2/20 0.42
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313370 0.93 KMT2A (0.42) ACHETDP1
SCHEMBL7823386 0.76 ADH1B (0.38) SMN1; SMN2MAPTHPGD
SCHEMBL7817328 0.76 ADH1B (0.38)
SCHEMBL7822809 0.75 CCR3 (0.37) SMN1; SMN2MAPTHPGD
SCHEMBL7827162 0.75 ADH1B (0.37)
Hydrochloric Acid SCHEMBL7463264 0.73 LMNA (0.46) SMN1; SMN2MAPT
SCHEMBL8313258 0.73 CHRM4 (0.56) CYP2D6
Hydrochloric Acid SCHEMBL7459792 0.73 CHRM4 (0.44) CYP2D6
SCHEMBL7468423 0.72 LMNA (0.46) SMN1; SMN2CYP2D6
SCHEMBL8315609 0.72 ADH1B (0.40) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0679642-B1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-11-10 EP disclosed
US-5654296-A HORMONE INHIBITOR; NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-08-05 US disclosed
US-5607939-A CALCIUM ANTAGONIST, GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONIST AND MONOAMINEU UPTAKE INHIBITORS FOR CENTRAL NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-04 US disclosed
EP-0679642-A1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-02 EP disclosed