SCHEMBL8313370

SCHEMBL8313370

O=CNCC(CCCN1C(=O)c2ccccc2C1=O)(c1ccccc1)c1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
ACHE P22303 8/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315366 0.93 ACHE (0.45) TDP1ACHE
SCHEMBL7816549 0.79 CCR3 (0.45) KMT2A
SCHEMBL7830286 0.79 KIF11 (0.39) KMT2A
SCHEMBL7459803 0.77 CHRM4 (0.50) DRD2DRD3
Hydrochloric Acid SCHEMBL7467316 0.76 CHRM4 (0.52) DRD2DRD3
Hydrochloric Acid SCHEMBL8869803 0.76 CHRM4 (0.52) DRD2DRD3
SCHEMBL7462064 0.75 MCHR1 (0.54) KMT2A
Hydrochloric Acid SCHEMBL7458878 0.75 MCHR1 (0.54) KMT2A
SCHEMBL7465175 0.75 DRD3 (0.51) TDP1DRD2DRD3
SCHEMBL7464640 0.74 MCHR1 (0.53) KMT2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0679642-B1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-11-10 EP disclosed
US-5654296-A HORMONE INHIBITOR; NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-08-05 US disclosed
US-5607939-A CALCIUM ANTAGONIST, GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONIST AND MONOAMINEU UPTAKE INHIBITORS FOR CENTRAL NERVOUS SYSTEM DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-04 US disclosed
EP-0679642-A1 Condensed heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-11-02 EP disclosed