SCHEMBL8315829

SCHEMBL8315829

CCc1cccc(Nc2ncnc3cnc(S(C)(=O)=O)nc23)c1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 17/20 0.51
PTGS1 P23219 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
GRM4 Q14833 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6990835 0.90 EGFR (0.50) EGFR
SCHEMBL6993872 0.85 EGFR (0.69) EGFR
SCHEMBL8314880 0.84 EGFR (0.53) EGFR
SCHEMBL8320084 0.84 EGFR (0.70) EGFR
SCHEMBL8315330 0.84 EGFR (0.57) EGFR
SCHEMBL6989584 0.84 EGFR (0.47) EGFRHDAC6
SCHEMBL6417047 0.84 EGFR (0.66) EGFR
SCHEMBL8320237 0.83 EGFR (0.55) EGFR
SCHEMBL8318188 0.82 EGFR (0.55) EGFR
SCHEMBL6994593 0.82 ABCG2 (0.54) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed