SCHEMBL8316860

SCHEMBL8316860

O=C1c2c(c3c4ccccc4[nH]c3c3[nH]c4ccccc4c23)C(=O)N1Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.70
CDK4 P11802 3/20 0.55
CCND1 P24385 3/20 0.55
PRKCA P17252 3/20 0.49
TACR1 P25103 1/20 0.48
CA9 Q16790 2/20 0.46
ATM Q13315 1/20 0.46
CA12 O43570 1/20 0.46
PARP14 Q460N5 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MAPT P10636 2/20 0.43
CCNE2 O96020 2/20 0.43
CCNE1 P24864 2/20 0.43
CDK2 P24941 2/20 0.43
CAMK2B Q13554 2/20 0.43
CAMK2G Q13555 2/20 0.43
CAMK2D Q13557 2/20 0.43
CAMK2A Q9UQM7 2/20 0.43
MEN1 O00255 1/20 0.43
PRKD3 O94806 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315890 0.88 NQO1 (0.53) NQO1CDK4CCND1TACR1CA9
SCHEMBL8313203 0.83 NQO1 (1.00) NQO1CDK4CCND1PRKCASMN1; SMN2
SCHEMBL14708720 0.81 NQO1 (0.64) NQO1CDK4CCND1PRKCACA9
SCHEMBL8318378 0.79 NQO1 (0.68) NQO1CDK4CCND1PRKCACA9
SCHEMBL8319736 0.79 CDK4 (0.47) NQO1CDK4CCND1PRKCASMN1; SMN2
SCHEMBL15959915 0.76 NQO1 (0.58) NQO1CDK4CCND1PRKCACA9
SCHEMBL18669003 0.75 CA9 (0.61) CA9ATMCA12SMN1; SMN2MAPT
SCHEMBL8324352 0.73 NQO1 (0.74) NQO1CDK4CCND1PRKCAMAPT
SCHEMBL8317087 0.72 ATM (0.58) CA9ATMCA12SMN1; SMN2MAPT
SCHEMBL14708729 0.72 NQO1 (0.49) NQO1CDK4CCND1PRKCAPARP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP claimed