SCHEMBL8313203

SCHEMBL8313203

O=C1c2c(c3c4ccccc4[nH]c3c3[nH]c4ccccc4c23)C(=O)N1Cc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 1.00
PRKCA P17252 5/20 0.61
CDK4 P11802 5/20 0.54
CCND1 P24385 5/20 0.54
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
CAMK2B Q13554 3/20 0.54
CAMK2G Q13555 3/20 0.54
CAMK2D Q13557 3/20 0.54
CAMK2A Q9UQM7 3/20 0.54
PRKD3 O94806 3/20 0.54
PRKCG P05129 3/20 0.54
PRKCB P05771 3/20 0.54
PRKACA P17612 3/20 0.54
PRKACG P22612 3/20 0.54
PRKACB P22694 3/20 0.54
PRKCH P24723 3/20 0.54
PRKCI P41743 3/20 0.54
PRKCE Q02156 3/20 0.54
PRKCQ Q04759 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324352 0.86 NQO1 (0.74) NQO1PRKCACDK4CCND1MEN1
SCHEMBL13431714 0.85 NQO1 (0.73) NQO1PRKCACDK4CCND1MAPT
SCHEMBL9623177 0.84 NQO1 (0.71) NQO1PRKCACDK4CCND1MEN1
SCHEMBL8316860 0.83 NQO1 (0.70) NQO1PRKCACDK4CCND1MEN1
SCHEMBL8318378 0.82 NQO1 (0.68) NQO1PRKCACDK4CCND1MEN1
SCHEMBL9622939 0.81 NQO1 (0.68) NQO1PRKCAMEN1KMT2AMAPT
SCHEMBL9622806 0.81 NQO1 (0.67) NQO1PRKCAMEN1KMT2AMAPT
SCHEMBL8314778 0.80 NQO1 (0.66) NQO1PRKCACDK4CCND1MEN1
SCHEMBL8312241 0.80 NQO1 (0.66) NQO1PRKCACDK4CCND1MEN1
SCHEMBL14708720 0.79 NQO1 (0.64) NQO1PRKCACDK4CCND1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP claimed
US-5547976-A VIRICIDES, HERPES VIRUS, CYTOMEGALOVIRUS; CARDIOVASCULAR DISORDERS BURROUGHS WELLCOME CO. (US) 1996-08-20 US claimed
EP-0630242-A1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1994-12-28 EP claimed
WO-1993018766-A1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1993-09-30 WO claimed
EP-0630242-B1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY WELLCOME FOUND (GB) 1999-01-20 EP disclosed
US-5547976-A VIRICIDES, HERPES VIRUS, CYTOMEGALOVIRUS; CARDIOVASCULAR DISORDERS BURROUGHS WELLCOME CO. (US) 1996-08-20 US disclosed
EP-0630242-A1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1994-12-28 EP disclosed
WO-1993018766-A1 FURTHER INDOLE DERIVATIVES WITH ANTIVIRAL ACTIVITY THE WELLCOME FOUNDATION LIMITED (GB) 1993-09-30 WO disclosed