SCHEMBL8317437

SCHEMBL8317437

ClCCCN1CCN(C(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 5/20 0.61
DRD2 P14416 4/20 0.61
P2RX7 Q99572 8/20 0.59
ADRA1B P35368 1/20 0.57
CHRM2 P08172 2/20 0.56
ADRA2A P08913 2/20 0.56
CYP2D6 P10635 2/20 0.56
HTR2A P28223 2/20 0.56
HRH1 P35367 2/20 0.56
HTR2B P41595 2/20 0.56
KCNH2 Q12809 2/20 0.56
CHRM4 P08173 1/20 0.56
CHRM5 P08912 1/20 0.56
ADORA3 P0DMS8 1/20 0.56
CHRM1 P11229 1/20 0.56
CHRM3 P20309 1/20 0.56
DRD1 P21728 1/20 0.56
ADRA1D P25100 1/20 0.56
HTR2C P28335 1/20 0.56
OPRM1 P35372 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28643710 0.98 DRD3 (0.59) DRD3DRD2P2RX7ADRA1BCHRM2
SCHEMBL7963339 0.90 DRD3 (0.59) DRD3DRD2P2RX7CHRM2ADRA2A
Hydrochloric Acid SCHEMBL8311562 0.88 DRD3 (0.58) DRD3DRD2P2RX7ADRA1BCHRM2
SCHEMBL7267063 0.84 ACHE (0.69) DRD3DRD2P2RX7ADRA1BCHRM2
SCHEMBL7670965 0.84 DRD3 (0.72) DRD3DRD2CHRM2ADRA2ACYP2D6
SCHEMBL11938950 0.83 OPRM1 (0.68) DRD3DRD2P2RX7ADRA1BCHRM2
SCHEMBL8051388 0.83 DRD3 (0.61) DRD3DRD2P2RX7ADRA1BCHRM2
SCHEMBL11206250 0.83 DRD3 (0.61) DRD3DRD2P2RX7ADRA1BCHRM2
SCHEMBL4249527 0.83 DRD3 (0.61) DRD3DRD2P2RX7ADRA1BCHRM2
SCHEMBL6618656 0.83 DRD3 (0.63) DRD3DRD2P2RX7ADRA1BCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7138236-A None JP disclosed
EP-3091001-B1 DIPHENYLMETHYL PIPERAZINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION USING SAME AETAS PHARMA CO LTD (JP) 2017-11-22 EP disclosed
EP-3091001-B1 DIPHENYLMETHYL PIPERAZINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION USING SAME AETAS PHARMA CO LTD (JP) 2017-11-22 EP disclosed
EP-3091001-A1 DIPHENYLMETHYL PIPERAZINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION USING SAME Aetas Pharma Co. Ltd. (JP) 2016-11-09 EP disclosed
EP-3091001-A1 DIPHENYLMETHYL PIPERAZINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION USING SAME Aetas Pharma Co. Ltd. (JP) 2016-11-09 EP disclosed
EP-2799430-B1 DIPHENYLMETHYL PIPERAZINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION USING SAME AETAS PHARMA CO LTD (JP) 2016-07-20 EP disclosed
EP-2799430-B1 DIPHENYLMETHYL PIPERAZINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION USING SAME AETAS PHARMA CO LTD (JP) 2016-07-20 EP disclosed
CN-103998428-B Diphenylmethyl piperazine derivatives and use the medical composition of this derivative AETAS PHARMA Co.,Ltd. (JP) 2016-03-23 CN disclosed
US-9073861-B2 Diphenylmethyl piperazine derivative and pharmaceutical composition using same AETAS PHARMA CO., LTD. (JP) 2015-07-07 US disclosed
US-9073861-B2 Diphenylmethyl piperazine derivative and pharmaceutical composition using same AETAS PHARMA CO., LTD. (JP) 2015-07-07 US disclosed
EP-0243905-A1 1-(omega-[bis-(phenyl)alkoxy]-alkyl)-4-(di-(phenyl)-methyl)piperazines, process for their preparation and medicines containing them Richter Gedeon Vegyészeti Gyár R.T. (HU) 1987-11-04 EP disclosed
EP-0115203-B1 BENZHYDRYLPIPERAZINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Richter Gedeon Vegyészeti Gyár R.T. (HU) 1987-04-01 EP disclosed
US-4504481-A ENZYME INHIBITORS IN LIVER TO REDUCE TOXIC EFFECT OF DRUGS RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1985-03-12 US disclosed
EP-0115203-A1 Benzhydrylpiperazine derivatives, process for their preparation and pharmaceutical compositions containing them Richter Gedeon Vegyészeti Gyár R.T. (HU) 1984-08-08 EP disclosed
US-4382934-A ANTIALLERGENS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-05-10 US disclosed
EP-0010398-B1 ISATIN DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1983-04-27 EP disclosed
EP-0006506-B1 CARBOSTYRILE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Roche Diagnostics GmbH (DE) 1981-09-16 EP disclosed
US-4234585-A ANTIALLERGENS, HYPOTENSIVE BOEHRINGER MANNHEIM GMBH (DE) 1980-11-18 US disclosed
EP-0010398-A1 Isatin derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1980-04-30 EP disclosed
EP-0006506-A1 Carbostyrile derivatives, processes for their preparation and pharmaceutical compositions containing them Roche Diagnostics GmbH (DE) 1980-01-09 EP disclosed