SCHEMBL8317449

SCHEMBL8317449

CC(Br)(c1ccccc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.67
TSHR P16473 1/20 0.67
KIF11 P52732 4/20 0.56
BACE1 P56817 1/20 0.47
TRPV6 Q9H1D0 2/20 0.47
CYP19A1 P11511 1/20 0.44
OPRM1 P35372 1/20 0.44
OPRL1 P41146 1/20 0.44
ESR1 P03372 2/20 0.41
ESR2 Q92731 2/20 0.41
CYP3A4 P08684 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MAPK1 P28482 1/20 0.41
ACP3 P15309 1/20 0.40
TACR1 P25103 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
ORAI1 Q96D31 1/20 0.38
ORAI2 Q96SN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoromethylbenzene SCHEMBL18787459 0.85 TSHR (0.82) ALDH1A1TSHRKIF11BACE1TRPV6
SCHEMBL134822 0.84 MAPK1 (0.52) ALDH1A1TSHRESR1ESR2CYP3A4
SCHEMBL17935746 0.83 ALDH1A1 (0.70) ALDH1A1TSHRKIF11BACE1TRPV6
Trifluoromethylbenzene SCHEMBL21879063 0.82 TSHR (0.88) ALDH1A1TSHRKIF11BACE1TRPV6
Trifluoromethylbenzene SCHEMBL4867878 0.82 TSHR (0.88) ALDH1A1TSHRKIF11BACE1TRPV6
Trifluoromethylbenzene SCHEMBL175647 0.82 TSHR (1.00) ALDH1A1TSHRKIF11BACE1TRPV6
Trifluoromethylbenzene SCHEMBL8692 0.82 TSHR (1.00) ALDH1A1TSHRKIF11BACE1TRPV6
Trifluoromethylbenzene SCHEMBL27760126 0.82 TSHR (1.00) ALDH1A1TSHRKIF11BACE1TRPV6
Trifluoromethylbenzene SCHEMBL11580827 0.79 TSHR (0.82) ALDH1A1TSHRKIF11BACE1TRPV6
Trifluoromethylbenzene SCHEMBL5311703 0.79 ALDH1A1 (0.82) ALDH1A1TSHRKIF11BACE1TRPV6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929534-A1 TRYCYCLIC COMPOUNDS AS PROSTAGLANDIN I2 RECEPTOR AGONISTS Takeda Pharmaceutical Company Limited (JP) 1999-07-21 EP disclosed
WO-1998013356-A1 TRYCYCLIC COMPOUNDS AS PROSTAGLANDIN I2 RECEPTOR AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-04-02 WO disclosed