SCHEMBL9733971

SCHEMBL9733971

NCC(Cc1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.50
SLC6A2 P23975 2/20 0.47
SLC6A4 P31645 2/20 0.47
SLC6A3 Q01959 2/20 0.47
KCNK2 O95069 1/20 0.47
KCNH2 Q12809 1/20 0.47
CACNA1C Q13936 1/20 0.47
TAAR1 Q96RJ0 1/20 0.46
SLC7A5 Q01650 4/20 0.43
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
GABBR2 O75899 1/20 0.42
GABBR1 Q9UBS5 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
PNMT P11086 1/20 0.41
ACP3 P15309 1/20 0.41
KIF11 P52732 1/20 0.41
MAOB P27338 1/20 0.41
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5178081 0.83 EPHX1 (0.47) KCNH2TAAR1GABBR2GABBR1ALDH1A1
SCHEMBL8810284 0.82 GABBR2 (0.53) SLC6A2SLC6A4SLC6A3TAAR1GABBR2
SCHEMBL1541691 0.82 GABBR2 (0.53) SLC6A2SLC6A4SLC6A3TAAR1GABBR2
SCHEMBL8621230 0.82 GABBR2 (0.53) SLC6A2SLC6A4SLC6A3TAAR1GABBR2
SCHEMBL9857073 0.81 SLC6A9 (0.57) SLC6A9SLC6A2SLC6A4SLC6A3KCNK2
Hydrochloric Acid SCHEMBL1983404 0.80 GABBR2 (0.52) SLC6A2SLC6A4SLC6A3TAAR1GABBR2
SCHEMBL11078290 0.78 TAAR1 (0.48) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL15903897 0.77 ESR1 (0.55) SLC6A2TAAR1SLC7A5GABBR2GABBR1
SCHEMBL5308356 0.77 CHRNB2 (0.54) SLC6A2SLC6A4SLC6A3TAAR1GABBR2
Hydrochloric Acid SCHEMBL9735324 0.77 CHRNB2 (0.55) TAAR1GABBR2GABBR1ALDH1A1ACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135955-A Anticoagulants or antifungal activity ELI LILLY AND COMPANY (US) 1992-08-04 US disclosed
EP-0339878-A2 Propanamine derivatives ELI LILLY AND COMPANY (US) 1989-11-02 EP disclosed