SCHEMBL8317467

SCHEMBL8317467

CCOC(=O)OC1C(C)CCCN1C(=O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
KMT2A Q03164 3/20 0.43
UTS2R Q9UKP6 1/20 0.43
SIGMAR1 Q99720 2/20 0.42
TSHR P16473 3/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
HPGD P15428 1/20 0.39
F2 P00734 1/20 0.39
POLB P06746 1/20 0.39
P2RX7 Q99572 1/20 0.39
ERCC1 P07992 1/20 0.39
ERCC4 Q92889 1/20 0.39
CCR3 P51677 1/20 0.38
CCR5 P51681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316830 0.94 KMT2A (0.43) ALDH1A1KMT2ASIGMAR1TSHRMEN1
SCHEMBL8315832 0.87 KMT2A (0.38) ALDH1A1KMT2AUTS2RTSHRMAPT
SCHEMBL9538321 0.85 SIGMAR1 (0.49) ALDH1A1KMT2AUTS2RSIGMAR1TSHR
SCHEMBL8316152 0.84 POLB (0.37) ALDH1A1KMT2AUTS2RMEN1LMNA
SCHEMBL8877185 0.84 ALDH1A1 (0.47) ALDH1A1KMT2AUTS2RSIGMAR1TSHR
SCHEMBL8317105 0.82 KMT2A (0.48) ALDH1A1KMT2ASIGMAR1TSHRMAPT
SCHEMBL8317694 0.82 KMT2A (0.43) ALDH1A1KMT2ASIGMAR1TSHRMEN1
SCHEMBL8316844 0.80 KMT2A (0.37) ALDH1A1KMT2ATSHRMEN1HPGD
SCHEMBL8316358 0.80 KMT2A (0.40) KMT2ASIGMAR1TSHRMEN1LMNA
SCHEMBL8318856 0.79 KMT2A (0.40) ALDH1A1KMT2ASIGMAR1TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501129-B1 Substituted bicyclic 3-arylpyrrolidin-2,4-dion derivatives BAYER AG (DE) 1999-07-14 EP disclosed
EP-0501129-A1 Substituted bicyclic 3-arylpyrrolidin-2,4-dion derivatives BAYER AG (DE) 1992-09-02 EP disclosed