SCHEMBL8317875

SCHEMBL8317875

O=C(O)c1ccc(NC(=O)c2cccc(Cl)c2Cl)cc1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.61
RAB9A P51151 3/20 0.61
JAK2 O60674 2/20 0.58
TSHR P16473 1/20 0.57
F2R P25116 1/20 0.56
MAOB P27338 1/20 0.56
JAK1 P23458 1/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
KCNK3 O14649 1/20 0.54
KCNK9 Q9NPC2 1/20 0.54
SMO Q99835 2/20 0.52
AVPR2 P30518 1/20 0.51
OXTR P30559 1/20 0.51
AVPR1A P37288 1/20 0.51
MAPT P10636 3/20 0.50
TP53 P04637 1/20 0.50
LCLAT1 Q6UWP7 1/20 0.49
ACLY P53396 1/20 0.49
PARP1 P09874 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12700230 0.86 ALDH1A1 (0.64) NPC1RAB9AMEN1KMT2AKCNK3
SCHEMBL27316696 0.82 AVPR2 (0.54) NPC1RAB9AMEN1KMT2AKCNK3
SCHEMBL8314314 0.82 AVPR2 (0.57) NPC1RAB9AMEN1KMT2AKCNK3
SCHEMBL7331517 0.81 DHODH (0.68) NPC1RAB9AMEN1KMT2AKCNK3
SCHEMBL4155586 0.81 JAK2 (0.73) NPC1RAB9AJAK2TSHRF2R
SCHEMBL7341264 0.80 TSHR (0.68) NPC1RAB9AJAK2TSHRJAK1
SCHEMBL15778670 0.80 FADS1 (0.68) NPC1RAB9AJAK2F2RMAOB
SCHEMBL1458777 0.80 CHRNB2 (0.63) TSHRMEN1KMT2ASMOAVPR2
SCHEMBL7334964 0.80 AVPR2 (0.57) NPC1RAB9AMEN1KMT2AAVPR2
SCHEMBL15779480 0.79 RAB9A (0.61) NPC1RAB9AJAK2F2RMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636625-B1 Tricyclic diazepines vasopressin and oxytocin antagonists AMERICAN CYANAMID CO (US) 1999-01-27 EP disclosed