SCHEMBL8318264

SCHEMBL8318264

O=C(O)CC1CCC(N2CCN(CCCNc3ccccn3)CC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.47
ADRA1A P35348 6/20 0.47
DRD3 P35462 6/20 0.47
ITGB3 P05106 5/20 0.46
ITGAV P06756 5/20 0.46
ITGB1 P05556 2/20 0.46
ITGA2B P08514 2/20 0.43
DPP4 P27487 1/20 0.41
ITGB5 P18084 1/20 0.41
TRPV6 Q9H1D0 1/20 0.40
GRIN2B Q13224 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300507 0.82 KDM4E (0.43) ITGB3ITGA2BTRPV6
SCHEMBL2843026 0.80 DRD3 (0.56) DRD2ADRA1ADRD3ITGB3ITGAV
SCHEMBL8304879 0.79 KDM4E (0.42) DRD2DRD3ITGB3ITGA2BTRPV6
SCHEMBL8304380 0.77 DRD3 (0.36) DRD2DRD3TRPV6
SCHEMBL8300030 0.75 KDM4E (0.45) DRD2ITGB3ITGA2BTRPV6GRIN2B
Trifluoroacetic Acid SCHEMBL5856786 0.74 DRD2 (0.53) DRD2ADRA1ADRD3ITGB3ITGAV
SCHEMBL7675724 0.74 DRD2 (0.49) DRD2ADRA1ADRD3ITGB3ITGAV
SCHEMBL4777735 0.74 CCR3 (0.56) GRIN2B
SCHEMBL13118499 0.73 DRD2 (0.61) DRD2ADRA1ADRD3
SCHEMBL8305139 0.73 CDK9 (0.36) DRD2TRPV6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906103-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-04-07 EP claimed
EP-0906103-A4 1999-04-07 EP claimed
WO-1997024124-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO claimed