SCHEMBL8304380

SCHEMBL8304380

O=C(O)CC1CCC(N2CCN(CCCCNc3ccnnc3)CC2)CC1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.36
DRD2 P14416 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CCNT1 O60563 2/20 0.34
CDK9 P50750 2/20 0.34
TRPV6 Q9H1D0 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
CCR3 P51677 1/20 0.34
HTR1A P08908 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305139 0.93 CDK9 (0.36) DRD2SMN1; SMN2CYP1A2CYP2D6CCNT1
SCHEMBL8304879 0.89 KDM4E (0.42) DRD3DRD2SMN1; SMN2CYP1A2CYP2D6
SCHEMBL8300507 0.85 KDM4E (0.43) SMN1; SMN2CYP1A2CYP2D6TRPV6KDM4E
SCHEMBL8305658 0.83 CCNT1 (0.38) CCNT1CDK9HTR2A
SCHEMBL8300030 0.81 KDM4E (0.45) DRD2CYP2D6CCNT1CDK9TRPV6
SCHEMBL8298648 0.80 CDK9 (0.36) CCNT1CDK9TRPV6KDM4EMEN1
SCHEMBL8318264 0.77 DRD2 (0.47) DRD3DRD2TRPV6
SCHEMBL8300003 0.77 CCR3 (0.39) CYP2D6CCR3
SCHEMBL8300686 0.75 NAMPT (0.43) CYP2D6CCNT1CDK9TRPV6KDM4E
SCHEMBL8300679 0.73 CCR3 (0.39) CYP2D6CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed