SCHEMBL8318325

SCHEMBL8318325

CCOC(=O)OC1C(C)C(C)C(C)N1C(=O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.39
LMNA P02545 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ERCC1 P07992 1/20 0.39
ERCC4 Q92889 1/20 0.39
CYP2C9 P11712 2/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
DPP4 P27487 1/20 0.36
P2RX7 Q99572 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
RECQL P46063 1/20 0.35
HTT P42858 1/20 0.35
ADCY8 P40145 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318132 0.85 ABCB1 (0.33) KMT2ALMNASMN1; SMN2CYP3A4GAA
SCHEMBL8316358 0.83 KMT2A (0.40) KMT2ALMNASMN1; SMN2ERCC1ERCC4
SCHEMBL8315566 0.82 SMN1; SMN2 (0.39) KMT2ALMNASMN1; SMN2CYP2C9CYP3A4
SCHEMBL8876339 0.82 KMT2A (0.41) KMT2ALMNASMN1; SMN2ERCC1ERCC4
SCHEMBL8316663 0.81 KMT2A (0.43) KMT2ALMNASMN1; SMN2CYP2C9CYP3A4
SCHEMBL8318855 0.81 KMT2A (0.40) KMT2ALMNASMN1; SMN2ERCC1ERCC4
SCHEMBL8313154 0.80 KMT2A (0.41) KMT2ALMNASMN1; SMN2ERCC1ERCC4
SCHEMBL8316830 0.79 KMT2A (0.43) KMT2ALMNASMN1; SMN2ERCC1ERCC4
SCHEMBL8312715 0.78 KMT2A (0.40) KMT2ALMNASMN1; SMN2ERCC1ERCC4
SCHEMBL8316915 0.78 TSHR (0.46) KMT2ALMNASMN1; SMN2TSHRSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501129-B1 Substituted bicyclic 3-arylpyrrolidin-2,4-dion derivatives BAYER AG (DE) 1999-07-14 EP disclosed
EP-0501129-A1 Substituted bicyclic 3-arylpyrrolidin-2,4-dion derivatives BAYER AG (DE) 1992-09-02 EP disclosed