SCHEMBL8318908

SCHEMBL8318908

O=C(/C=C/c1cccc(Cn2cnc(-c3ccccc3)c2)c1)NOC1CCCCO1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
KDM1A O60341 1/20 0.39
HDAC1 Q13547 9/20 0.39
HDAC8 Q9BY41 9/20 0.39
HDAC6 Q9UBN7 9/20 0.39
TBXAS1 P24557 1/20 0.38
BCHE P06276 2/20 0.38
ACHE P22303 2/20 0.38
TGFBR1 P36897 1/20 0.38
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
HDAC4 P56524 1/20 0.37
MEF2D Q14814 1/20 0.37
MGLL Q99685 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323958 0.80 HDAC1 (0.40) HDAC1HDAC8HDAC6TGFBR1HDAC4
SCHEMBL8325909 0.80 HDAC4 (0.55) KDM4AKDM4CHDAC1HDAC8HDAC6
SCHEMBL1579332 0.79 NPSR1 (0.43) HDAC1HDAC8HDAC6TGFBR1HDAC4
SCHEMBL1579334 0.79 NPSR1 (0.43) HDAC1HDAC8HDAC6TGFBR1HDAC4
SCHEMBL1164811 0.78 HDAC1 (0.37) HDAC1HDAC8HDAC6BCHEACHE
SCHEMBL3439472 0.78 HDAC1 (0.37) HDAC1HDAC8HDAC6BCHEACHE
SCHEMBL8319569 0.78 TGFBR1 (0.44) HDAC1HDAC8HDAC6TGFBR1HDAC4
SCHEMBL8318730 0.77 TBXAS1 (0.60) KDM4AKDM4CTBXAS1CYP2E1CYP3A4
SCHEMBL4258903 0.77 MGLL (0.46) HDAC1HDAC8HDAC6HDAC4MGLL
SCHEMBL4258906 0.77 MGLL (0.46) HDAC1HDAC8HDAC6HDAC4MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed