SCHEMBL8325909

SCHEMBL8325909

O=C(/C=C/c1cccc(Cn2cnc(-c3ccccc3)c2)c1)NO

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.55
MEF2D Q14814 2/20 0.55
HDAC1 Q13547 13/20 0.54
HDAC8 Q9BY41 12/20 0.54
HDAC6 Q9UBN7 11/20 0.54
TBXAS1 P24557 1/20 0.50
KDM4A O75164 1/20 0.49
KDM4C Q9H3R0 1/20 0.49
CYP2E1 P05181 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2A6 P11509 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2B6 P20813 1/20 0.49
CYP2C19 P33261 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC2 Q92769 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318730 0.91 TBXAS1 (0.60) TBXAS1KDM4AKDM4CCYP2E1CYP3A4
SCHEMBL8326744 0.90 HDAC1 (0.56) HDAC4HDAC1HDAC8HDAC6CYP2E1
SCHEMBL8325813 0.82 TBXAS1 (0.56) HDAC4HDAC1HDAC8HDAC6TBXAS1
SCHEMBL8319688 0.82 TBXAS1 (0.46) HDAC1HDAC8HDAC6TBXAS1KDM4A
SCHEMBL1165168 0.81 HDAC1 (0.61) HDAC4MEF2DHDAC1HDAC8HDAC6
SCHEMBL1165170 0.81 HDAC1 (0.61) HDAC4MEF2DHDAC1HDAC8HDAC6
SCHEMBL8318908 0.80 KDM4A (0.40) HDAC4MEF2DHDAC1HDAC8HDAC6
SCHEMBL8322937 0.78 CYP3A4 (0.49) HDAC1HDAC8TBXAS1KDM4AKDM4C
SCHEMBL13762662 0.75 HDAC4 (0.71) HDAC4MEF2DHDAC1HDAC8HDAC6
SCHEMBL13762664 0.75 HDAC4 (0.71) HDAC4MEF2DHDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed