SCHEMBL8318934

SCHEMBL8318934

O=C(O)c1ccc(CCc2ccccc2OCc2ccccc2)cc1O

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.60
DRD2 P14416 4/20 0.60
PTGER1 P34995 1/20 0.56
PTGER4 P35408 1/20 0.56
PTGER3 P43115 1/20 0.56
PTGER2 P43116 1/20 0.56
ABCB1 P08183 9/20 0.54
MCL1 Q07820 1/20 0.52
ABCG2 Q9UNQ0 1/20 0.51
FOLH1 Q04609 2/20 0.50
MAOB P27338 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8409730 0.95 HTR1A (0.60) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8319789 0.93 PTGER1 (0.67) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8319729 0.88 ABCB1 (0.56) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8321056 0.87 FOLH1 (0.51) PTGER1FOLH1
SCHEMBL8326478 0.87 PTGER1 (0.57) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8318400 0.85 ABCB1 (0.65) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL8319605 0.85 MTNR1A (0.58) HTR1ADRD2ABCB1MAOB
SCHEMBL8322796 0.84 GCK (0.47) HTR1ADRD2PTGER1PTGER4PTGER3
SCHEMBL6261880 0.83 PPARA (0.55) MCL1
SCHEMBL8324057 0.81 PTGER4 (0.59) HTR1ADRD2PTGER1PTGER4PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP claimed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP claimed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO claimed
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed