SCHEMBL8319666

SCHEMBL8319666

CCCCc1ncc(C[C@H](N)C(=O)O)[nH]1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.48
SLC7A5 Q01650 1/20 0.48
GRM5 P41594 1/20 0.46
BRS3 P32247 3/20 0.46
CYP1A2 P05177 1/20 0.41
RECQL P46063 1/20 0.41
SLC1A3 P43003 1/20 0.40
KIF11 P52732 1/20 0.40
GRIA1 P42261 1/20 0.38
GRIA2 P42262 1/20 0.38
GRIA3 P42263 1/20 0.38
GRIA4 P48058 1/20 0.38
KDM6B O15054 1/20 0.38
KDM4A O75164 1/20 0.38
KDM4D Q6B0I6 1/20 0.38
KDM3B Q7LBC6 1/20 0.38
HIF1AN Q9NWT6 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
KDM2A Q9Y2K7 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29356218 0.89 SLC7A5 (0.51) CYP3A4SLC7A5CYP1A2RECQLSLC1A3
Methylamine SCHEMBL29022748 0.86 CYP3A4 (0.46) CYP3A4SLC7A5GRM5SLC1A3GRIA1
SCHEMBL849758 0.83 SLC7A5 (0.51) CYP3A4SLC7A5CYP1A2SLC1A3GRIA1
SCHEMBL20539892 0.82 ARG2 (0.46) CYP3A4SLC7A5SLC1A3GRIA1GRIA2
SCHEMBL29022740 0.81 SLC7A5 (0.47) CYP3A4SLC7A5BRS3SLC1A3GRIA1
SCHEMBL27446953 0.80 SLC7A5 (0.51) CYP3A4SLC7A5CYP1A2RECQLSLC1A3
SCHEMBL8326405 0.79 BRS3 (0.42) BRS3
SCHEMBL5292853 0.78 SLC7A5 (0.53) CYP3A4SLC7A5CYP1A2SLC1A3GRIA1
SCHEMBL1539194 0.78 SLC7A5 (0.53) CYP3A4SLC7A5CYP1A2SLC1A3GRIA1
SCHEMBL26912795 0.78 SLC7A5 (0.53) CYP3A4SLC7A5CYP1A2SLC1A3GRIA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0589665-B1 4,5,6,7-Tetrahydro-1H-imidazo 4,5-c pyridine-6-carboxylic acid amide derivatives as angiotensine II antagonistes KUREHA CHEMICAL IND CO LTD (JP) 1999-11-17 EP disclosed
US-5401736-A Angiotensis II antagonists KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1995-03-28 US disclosed
EP-0589665-A2 4,5,6,7-Tetrahydro-1H-imidazo 4,5-c pyridine-6-carboxylic acid amide derivatives as angiotensine II antagonistes KUREHA KAGAKU KOGYO KABUSHIKI KAISHA (JP) 1994-03-30 EP disclosed