SCHEMBL8320059

SCHEMBL8320059

CS(=O)(=O)O.C[Si](C)(C)Oc1ccc(-c2cccc(S)c2-c2ccc(O[Si](C)(C)C)cc2)cc1

nearest known ligand 0.33

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.33
PPARA Q07869 4/20 0.33
HDAC4 P56524 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
ENPP1 P22413 1/20 0.32
PTGS2 P35354 5/20 0.32
PTGS1 P23219 1/20 0.31
JAK2 O60674 1/20 0.31
JAK3 P52333 1/20 0.31
PTK2 Q05397 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322919 0.84 ADORA2A (0.37) HSP90AA1HSP90AB1
SCHEMBL8320148 0.81 PPARA (0.39) PPARGPPARAHDAC4HDAC2HDAC8
SCHEMBL8322203 0.77 PPARA (0.36) PPARGPPARAHSP90AA1
SCHEMBL8323471 0.76 ELANE (0.48) PPARGPPARAHSP90AA1HSP90AB1
SCHEMBL8322952 0.76 ENPP1 (0.35) PPARGPPARAHDAC4HDAC2HDAC8
SCHEMBL8323062 0.75 OXTR (0.39)
Trifluoromethanesulfonic Acid SCHEMBL3143639 0.75 ENPP1 (0.46) HDAC4HDAC2HDAC8HSP90AA1HSP90AB1
SCHEMBL8648344 0.74 PTGS2 (0.38) PTGS2PTGS1
SCHEMBL8317959 0.74 OXTR (0.36) PPARGPPARAHSP90AA1HSP90AB1
Sulfuric Acid SCHEMBL15345275 0.74 PPARG (0.37) PPARGPPARAHDAC4HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5880169-A HAVING HIGH RESOLUTION FOR FINE PATTERNING SHIN-ETSU CHEMICAL CO., LTD. (JP) 1999-03-09 US disclosed