SCHEMBL8320127

SCHEMBL8320127

COc1cc(OC)nc(C2OC(=O)c3c(-c4ccccc4)ccnc32)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.37
HCRTR2 O43614 3/20 0.37
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
ALDH1A1 P00352 3/20 0.36
PGR P06401 1/20 0.36
IDO1 P14902 1/20 0.35
MAPT P10636 3/20 0.35
PKM P14618 2/20 0.35
KDM4E B2RXH2 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAOA P21397 2/20 0.34
MAOB P27338 2/20 0.33
LYN P07948 1/20 0.32
SRC P12931 1/20 0.32
BTK Q06187 1/20 0.32
HPGD P15428 1/20 0.32
PTPN7 P35236 1/20 0.32
BLM P54132 1/20 0.32
WRN Q14191 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319649 0.82 MAOB (0.39) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL8322076 0.68 HCRTR1 (0.36) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL8807990 0.68 ACHE (0.37) HCRTR1HCRTR2ALDH1A1KDM4ESMN1; SMN2
SCHEMBL8809644 0.67 NPSR1 (0.37) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL8321570 0.66 NPC1 (0.35) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL8323374 0.63 EDNRA (0.37) NPC1RAB9AALDH1A1MAPTMAOA
SCHEMBL9176204 0.62 HCRTR1 (0.42) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL28635180 0.62 KMT2A (0.50) NPC1RAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL744054 0.60 IDO1 (0.50) IDO1
SCHEMBL9180424 0.60 ALDH1A1 (0.45) HCRTR1HCRTR2ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0752424-B1 NICOTINIC ACID DERIVATIVE AND HERBICIDE KUMIAI CHEMICAL INDUSTRY CO (JP) 1999-06-16 EP disclosed
US-5877120-A Nicotinic acid derivatives and herbicides KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1999-03-02 US disclosed
EP-0752424-A1 NICOTINIC ACID DERIVATIVE AND HERBICIDE KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1997-01-08 EP disclosed