SCHEMBL8322110

SCHEMBL8322110

CC(C)(N)c1ccccc1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.47
SLC6A2 P23975 1/20 0.47
TAAR1 Q96RJ0 1/20 0.47
CALM1 P0DP23 1/20 0.42
BCL2 P10415 1/20 0.41
BCL2L1 Q07817 1/20 0.41
LTA4H P09960 1/20 0.40
HPGD P15428 2/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 1/20 0.39
CYP2D6 P10635 1/20 0.39
DRD2 P14416 1/20 0.38
DRD1 P21728 1/20 0.38
DRD4 P21917 1/20 0.38
DRD5 P21918 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ATM Q13315 1/20 0.38
HRH1 P35367 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL28430480 0.98 HTR2A (0.46) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL28662452 0.85 HTR2A (0.42) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL6546758 0.83 CALM1 (0.46) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL10782398 0.82 CALM1 (0.44) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL8815094 0.80 BCL2 (0.45) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL29470998 0.80 BCL2 (0.45) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL10900432 0.78 HTR2A (0.41) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL3435481 0.78 KCNN4 (0.50) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL10601601 0.78 LMNA (0.47) HTR2ASLC6A2TAAR1CALM1BCL2
SCHEMBL5764360 0.77 CALM1 (0.48) HTR2ACALM1BCL2BCL2L1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592684-B1 MALONAMIDE DERIVATIVES AS GAMMA-SECRETASE INHIBITORS HOFFMANN LA ROCHE (CH) 2008-07-30 EP disclosed
WO-2004069826-A1 MALONAMIDE DERIVATIVES AS GAMMA-SECRETASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-08-19 WO disclosed