SCHEMBL8322119

SCHEMBL8322119

CN(C)c1ccc([S+](c2ccc(OC3CCCCO3)cc2)c2ccc(N(C)C)cc2)cc1.CS(=O)(=O)[O-]

nearest known ligand 0.43

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 3/20 0.34
HSD11B1 P28845 1/20 0.33
HPGD P15428 2/20 0.32
NPC1 O15118 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TP53 P04637 2/20 0.32
MAPT P10636 1/20 0.32
TNK2 Q07912 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322269 0.97 GAA (0.36) DDB1CRBNKMT2AMEN1GAA
SCHEMBL8327555 0.92 DDB1 (0.36) DDB1CRBNKMT2AMEN1GAA
SCHEMBL6140565 0.91 ALDH1A1 (0.34) DDB1CRBNKMT2AMEN1GAA
SCHEMBL8663699 0.91 ALDH1A1 (0.34) DDB1CRBNKMT2AMEN1GAA
SCHEMBL8322230 0.90 DHFR (0.36) GAAHSD11B1ALDH1A1
SCHEMBL8651820 0.89 GAA (0.32) DDB1CRBNKMT2AMEN1GAA
SCHEMBL8325663 0.88 GAA (0.38) DDB1CRBNKMT2AMEN1GAA
SCHEMBL8317952 0.87 MEN1 (0.38) KMT2AMEN1HSD11B1NPC1SMN1; SMN2
SCHEMBL6140612 0.87 HPGD (0.37) KMT2AMEN1GAAHPGDNPC1
SCHEMBL8321358 0.86 GAA (0.35) KMT2AMEN1GAAHSD11B1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5880169-A HAVING HIGH RESOLUTION FOR FINE PATTERNING SHIN-ETSU CHEMICAL CO., LTD. (JP) 1999-03-09 US disclosed