SCHEMBL8322244

SCHEMBL8322244

CC(C)Oc1ccc(-c2nnn(C)n2)cc1C=O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACLY P53396 1/20 0.39
ERN1 O75460 2/20 0.38
S1PR1 P21453 1/20 0.36
S1PR5 Q9H228 1/20 0.36
SHMT2 P34897 1/20 0.35
LRRK2 Q5S007 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 1/20 0.34
NPC1 O15118 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34
XDH P47989 1/20 0.34
POLB P06746 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5190700 0.85 ACLY (0.48) ACLYERN1LRRK2SMN1; SMN2MAPT
SCHEMBL8328118 0.77 ALDH1A1 (0.42) ACLYERN1S1PR1LRRK2SMN1; SMN2
SCHEMBL8322837 0.74 ALDH1A1 (0.56) ERN1MAPTMEN1ALDH1A1KMT2A
SCHEMBL12896173 0.73 NPC1 (0.50) SMN1; SMN2MAPTNPC1NFKB1RAB9A
SCHEMBL13846196 0.71 MAPT (0.60) ACLYLRRK2SMN1; SMN2MAPTMEN1
SCHEMBL6097515 0.71 ERN1 (0.51) ERN1MAPTMEN1ALDH1A1KMT2A
SCHEMBL8329005 0.70 ERN1 (0.39) ERN1S1PR1MAPTMEN1ALDH1A1
SCHEMBL6264 0.70 SMN1; SMN2 (0.43) SMN1; SMN2NPC1NFKB1RAB9ANFKB2
SCHEMBL6098469 0.69 ERN1 (0.45) ACLYERN1MAPTMEN1ALDH1A1
SCHEMBL18004001 0.68 XDH (0.43) ERN1XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858444-A4 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1999-12-01 EP disclosed
EP-0858444-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-08-19 EP disclosed
US-5750549-A ANTIINFLAMMATORY AGENTS OR ANALGESICS MERCK & CO., INC. (US) 1998-05-12 US disclosed
WO-1997014671-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-04-24 WO disclosed