SCHEMBL8319903

SCHEMBL8319903

Oc1c2ncc3cccc(F)c3c2nn1-c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 5/20 0.37
GABRA2 P47869 5/20 0.37
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PARP1 P09874 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
PARP3 Q9Y6F1 1/20 0.33
SLC40A1 Q9NP59 1/20 0.33
RARG P13631 1/20 0.33
RORC P51449 1/20 0.33
KDM4E B2RXH2 1/20 0.32
SCN9A Q15858 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322376 0.79 SMN1; SMN2 (0.49) GABRA1GABRA2NPC1LMNARAB9A
SCHEMBL8468606 0.78 NPC1 (0.40) GABRA1GABRA2TP53POLBRXFP1
Water SCHEMBL8323447 0.67 LMNA (0.37) TP53RXFP1LMNARAB9ASMN1; SMN2
SCHEMBL8321754 0.66 KDM4E (0.41) TP53POLBLMNASMN1; SMN2KDM4E
SCHEMBL8320446 0.66 NPC1 (0.49) GABRA1GABRA2NPC1LMNARAB9A
SCHEMBL8466300 0.66 GAA (0.43) TP53POLBNPC1LMNARAB9A
SCHEMBL8466029 0.64 SCN9A (0.32) NPC1LMNARAB9ASMN1; SMN2KDM4E
SCHEMBL8329043 0.63 TEAD1 (0.39) TP53SMN1; SMN2
SCHEMBL8322673 0.63 AURKA (0.36) TP53POLBNPC1LMNARAB9A
SCHEMBL8523787 0.63 NPC1 (0.52) GABRA1GABRA2NPC1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888347-A1 PHARMACEUTICALLY USEFUL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-01-07 EP claimed
WO-1997034893-A1 PHARMACEUTICALLY USEFUL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-09-25 WO claimed