SCHEMBL8322601

SCHEMBL8322601

COC(c1ccccc1)n1c(=O)c2ccccc2c2nn(-c3ccc(C(F)(F)F)cc3)c(O)c21

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CASR P41180 2/20 0.39
SYK P43405 1/20 0.38
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
TRPV1 Q8NER1 1/20 0.34
HIF1A Q16665 1/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
KMT2A Q03164 1/20 0.34
TRPV4 Q9HBA0 1/20 0.34
ADORA1 P30542 1/20 0.34
MPI P34949 1/20 0.34
PHOSPHO1 Q8TCT1 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CXCR3 P49682 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8320581 0.79 NPSR1 (0.48) NPSR1KDM4ESYKLMNAALDH1A1
SCHEMBL8322607 0.73 MEN1 (0.43) NPSR1KDM4EALDH1A1TRPV1MEN1
SCHEMBL8324351 0.73 MAPT (0.46) KDM4ELMNAALDH1A1MEN1MAPT
SCHEMBL8460257 0.70 NPSR1 (0.46) NPSR1KDM4ECASRSYKLMNA
SCHEMBL8321791 0.70 L3MBTL1 (0.39) NPSR1KDM4ESYKALDH1A1TRPV1
SCHEMBL8462289 0.70 MAPT (0.47) NPSR1KDM4ESYKTRPV1HIF1A
SCHEMBL8522571 0.68 ADORA3 (0.47) NPSR1KDM4ESYKTRPV1HIF1A
SCHEMBL8523766 0.66 KDM4E (0.39) KDM4ELMNAALDH1A1MEN1MAPT
Water SCHEMBL8326580 0.66 MAPT (0.38) NPSR1KDM4ESYKTRPV1HIF1A
SCHEMBL8328108 0.65 MAPT (0.40) NPSR1KDM4ESYKTRPV1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888347-A1 PHARMACEUTICALLY USEFUL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-01-07 EP disclosed
WO-1997034893-A1 PHARMACEUTICALLY USEFUL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-09-25 WO disclosed