SCHEMBL8322773

SCHEMBL8322773

Cc1cn(Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)c2c(C(=O)O)cccc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.46
ABCB11 O95342 1/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
CYP3A4 P08684 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
CYP2C9 P11712 1/20 0.40
ADRB3 P13945 1/20 0.40
ADRA2B P18089 1/20 0.40
SLC6A2 P23975 1/20 0.40
TBXAS1 P24557 1/20 0.40
HTR2C P28335 1/20 0.40
AGTR1 P30556 1/20 0.40
PPARG P37231 1/20 0.40
HTR2B P41595 1/20 0.40
AGTR2 P50052 1/20 0.40
PDE3A Q14432 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328346 0.92 CHRM1 (0.55) CHRM1
SCHEMBL8325881 0.90 CHRM1 (0.45) CHRM1ABCB11EGFRERBB2CYP3A4
SCHEMBL8323834 0.87 CHRM1 (0.40) CHRM1ABCB11EGFRERBB2CYP3A4
SCHEMBL8329298 0.87 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL4729358 0.79 ABCB11 (0.47) ABCB11EGFRERBB2CYP3A4ADORA3
SCHEMBL8328347 0.79 CHRM1 (0.41) CHRM1ABCB11EGFRERBB2CYP3A4
SCHEMBL8325882 0.78 CHRM1 (0.39) CHRM1ABCB11EGFRERBB2CYP3A4
SCHEMBL7006258 0.78 ABCB11 (0.47) ABCB11EGFRERBB2CYP3A4ADORA3
SCHEMBL9197386 0.78 ABCB11 (0.56) ABCB11EGFRERBB2CYP3A4ADORA3
SCHEMBL7007755 0.77 AGTR1 (0.49) AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0498721-B1 N-substituted quinoline derivatives, process for their preparation, their use as pharmaceuticals and pharmaceutical compositions containing them HOECHST MARION ROUSSEL INC (FR) 1999-12-22 EP claimed
US-5985894-A USEFUL IN THE TREATMENT OF CARDIOVASCULAR ILLNESSES HOECHST MARION ROUSSEL (FR) 1999-11-16 US disclosed