SCHEMBL8322947

SCHEMBL8322947

O=c1[nH]c2c(c(=O)n1Cc1ccccc1)CN(Cc1ccccc1)CC2

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.67
ACHE P22303 3/20 0.60
GABRA1 P14867 4/20 0.58
GABRA2 P47869 4/20 0.58
CLPP Q16740 1/20 0.56
SLC6A5 Q9Y345 1/20 0.55
GABRA5 P31644 2/20 0.53
GABRA3 P34903 2/20 0.53
AKR1B1 P15121 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8323565 0.99 HPGD (0.65) HPGDACHEGABRA1GABRA2CLPP
SCHEMBL22028762 0.94 CLPP (0.60) HPGDACHEGABRA1GABRA2CLPP
SCHEMBL22071231 0.93 KDM4E (0.62) HPGDACHEGABRA1GABRA2CLPP
SCHEMBL22028736 0.90 CLPP (0.62) HPGDACHEGABRA1GABRA2CLPP
SCHEMBL22028733 0.90 ACHE (0.58) HPGDACHEGABRA1GABRA2CLPP
SCHEMBL8323169 0.87 ACHE (0.57) ACHEGABRA1GABRA2SLC6A5GABRA5
Hydrochloric Acid SCHEMBL8323662 0.86 ACHE (0.56) ACHEGABRA1GABRA2SLC6A5GABRA5
Hydrochloric Acid SCHEMBL8323549 0.84 HPGD (0.64) HPGDACHEGABRA1GABRA2CLPP
SCHEMBL8324851 0.80 ACHE (0.55) ACHEGABRA1GABRA2SLC6A5GABRA5
SCHEMBL2625346 0.80 SLC6A5 (0.80) ACHEGABRA1GABRA2CLPPSLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0621037-B1 Pyrido-pyrimidinediones, process for their preparation and their use as pharmaceuticals HOECHST AG (DE) 1999-07-07 EP disclosed
US-5556854-A CARDIOVASCULAR DISORDERS AND/OR NEUROGENERATIVE DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1996-09-17 US disclosed
EP-0621037-A1 Pyrido-pyrimidinediones, process for their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1994-10-26 EP disclosed