SCHEMBL8323169

SCHEMBL8323169

Cn1c(=O)[nH]c2c(c1=O)CN(Cc1ccccc1)CC2

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.57
GABRA1 P14867 5/20 0.56
GABRA2 P47869 5/20 0.56
GABRA5 P31644 2/20 0.54
GABRA3 P34903 2/20 0.54
SLC6A5 Q9Y345 1/20 0.53
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8323662 0.99 ACHE (0.56) ACHEGABRA1GABRA2GABRA5GABRA3
SCHEMBL8324851 0.88 ACHE (0.55) ACHEGABRA1GABRA2GABRA5GABRA3
SCHEMBL8322947 0.87 HPGD (0.67) ACHEGABRA1GABRA2GABRA5GABRA3
Hydrochloric Acid SCHEMBL8323565 0.86 HPGD (0.65) ACHEGABRA1GABRA2GABRA5GABRA3
SCHEMBL22071231 0.83 KDM4E (0.62) ACHEGABRA1GABRA2GABRA5GABRA3
SCHEMBL2303143 0.82 ACHE (0.53) ACHEGABRA1GABRA2GABRA5GABRA3
SCHEMBL22028762 0.81 CLPP (0.60) ACHEGABRA1GABRA2GABRA5GABRA3
SCHEMBL22028733 0.80 ACHE (0.58) ACHEGABRA1GABRA2GABRA5GABRA3
SCHEMBL8319246 0.80 SLC6A5 (0.56) ACHEGABRA1GABRA2SLC6A5KDM4E
SCHEMBL8319661 0.79 CLPP (0.54) ACHEKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0621037-B1 Pyrido-pyrimidinediones, process for their preparation and their use as pharmaceuticals HOECHST AG (DE) 1999-07-07 EP disclosed
US-5556854-A CARDIOVASCULAR DISORDERS AND/OR NEUROGENERATIVE DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1996-09-17 US disclosed
EP-0621037-A1 Pyrido-pyrimidinediones, process for their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1994-10-26 EP disclosed