SCHEMBL8323908

SCHEMBL8323908

CSc1c(C#N)c(=O)n(C)c(=O)n1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
KDM4E B2RXH2 5/20 0.48
LMNA P02545 1/20 0.48
MAPK1 P28482 1/20 0.44
PGR P06401 1/20 0.43
GRIA2 P42262 1/20 0.43
GRIA4 P48058 1/20 0.43
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
EGFR P00533 1/20 0.40
SRC P12931 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
KCNJ5 P48544 1/20 0.38
KCNJ3 P48549 1/20 0.38
KCNQ1 P51787 1/20 0.38
CACNA1C Q13936 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328828 0.76 AOC3 (0.45) ALDH1A1L3MBTL1KDM4ELMNAMAPK1
SCHEMBL8327964 0.72 GRIA2 (0.39) ALDH1A1L3MBTL1KDM4ELMNAMAPK1
SCHEMBL8327668 0.71 GRIA2 (0.41) ALDH1A1L3MBTL1KDM4ELMNAMAPK1
SCHEMBL9710841 0.70 GSK3B (0.50) ALDH1A1KDM4ELMNAMAPK1PGR
SCHEMBL8328438 0.70 ALDH1A1 (0.38) ALDH1A1L3MBTL1KDM4EMAPK1GRIA2
SCHEMBL8328148 0.69 GRIA4 (0.41) ALDH1A1L3MBTL1KDM4ELMNAMAPK1
SCHEMBL8328146 0.69 GRIA4 (0.41) ALDH1A1L3MBTL1KDM4ELMNAMAPK1
SCHEMBL8326586 0.67 ALDH1A1 (0.40) ALDH1A1L3MBTL1KDM4ELMNAMAPK1
SCHEMBL9710619 0.67 GSK3B (0.46) ALDH1A1KDM4EMAPK1PGRGSK3A
SCHEMBL9711058 0.67 KDM4E (0.48) ALDH1A1L3MBTL1KDM4ELMNAGRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed