SCHEMBL8326586

SCHEMBL8326586

CSc1c(C#N)c(=O)n(C)c(=S)n1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 7/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GRIA2 P42262 2/20 0.38
GRIA4 P48058 2/20 0.38
NPC1 O15118 1/20 0.36
CRHBP P24387 1/20 0.36
RAB9A P51151 1/20 0.36
CRHR2 Q13324 1/20 0.36
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP1 P29466 1/20 0.34
HSD17B10 Q99714 1/20 0.34
EGFR P00533 1/20 0.33
SRC P12931 1/20 0.33
AOC3 Q16853 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328828 0.81 AOC3 (0.45) ALDH1A1L3MBTL1KDM4ELMNAMAPT
SCHEMBL8327686 0.79 GRIA2 (0.35) GRIA2GRIA4EGFRSRC
SCHEMBL8329433 0.71 GRIA2 (0.36) GRIA2GRIA4
SCHEMBL8329429 0.71 GRIA2 (0.36) GRIA2GRIA4
SCHEMBL18656052 0.71 LPO (0.32)
SCHEMBL24380727 0.63 ALDH1A1 (0.60) ALDH1A1L3MBTL1KDM4ELMNAMAPT
SCHEMBL16402408 0.63 GAA (0.39) ALDH1A1L3MBTL1KDM4ELMNAMEN1
SCHEMBL19486386 0.62
SCHEMBL15700494 0.59 KDM4E (0.49) ALDH1A1L3MBTL1KDM4ELMNAMAPT
SCHEMBL2760401 0.59 KDM4E (0.44) ALDH1A1L3MBTL1KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed