SCHEMBL8322760

SCHEMBL8322760

CC(C)(C)c1cnc(Cc2ccc(/C=C/C(=O)O)cc2)[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 4/20 0.48
BRS3 P32247 1/20 0.45
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MITF O75030 1/20 0.44
KLF5 Q13887 1/20 0.44
CYP26A1 O43174 1/20 0.43
CYP26B1 Q9NR63 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
NPC1 O15118 1/20 0.42
CASP3 P42574 1/20 0.42
RAB9A P51151 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MAPK1 P28482 1/20 0.41
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323151 0.88 HDAC1 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8324028 0.86 NR1H4 (0.40) TBXAS1BRS3HDAC3HDAC4HDAC1
SCHEMBL8319501 0.75 THRB (0.54) TBXAS1BRS3KDM4EALDH1A1HPGD
SCHEMBL8322805 0.74 BRS3 (0.48) TBXAS1BRS3KDM4EALDH1A1HPGD
SCHEMBL8324034 0.73 RECQL (0.45) TBXAS1BRS3KDM4EALDH1A1HPGD
SCHEMBL8921111 0.72 TBXAS1 (0.68) TBXAS1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL9401700 0.72 TAAR1 (0.55) TBXAS1KDM4EALDH1A1HPGDSMN1; SMN2
SCHEMBL9507338 0.72 TAAR1 (0.55) TBXAS1KDM4EALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL7266355 0.71 TBXAS1 (0.54) TBXAS1KDM4EALDH1A1HPGDSMN1; SMN2
Hydrochloric Acid SCHEMBL11261045 0.70 TBXAS1 (0.53) TBXAS1KDM4EALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed