SCHEMBL8324034

SCHEMBL8324034

COc1ccccc1-c1cnc(Cc2ccc(/C=C/C(=O)O)cc2)[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.45
TBXAS1 P24557 2/20 0.44
AKR1C3 P42330 1/20 0.43
BRS3 P32247 1/20 0.41
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ESR1 P03372 2/20 0.41
THRB P10828 1/20 0.40
ATM Q13315 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
SNCA P37840 2/20 0.39
CA2 P00918 2/20 0.39
CA5A P35218 2/20 0.39
CA9 Q16790 2/20 0.39
CA12 O43570 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323117 0.90 HDAC1 (0.52) HDAC3HDAC1HDAC2HDAC8HDAC4
SCHEMBL8323886 0.87 NR1H4 (0.40) BRS3ESR1ABCG2HDAC3HDAC1
SCHEMBL8319501 0.81 THRB (0.54) TBXAS1AKR1C3BRS3KDM4EALDH1A1
SCHEMBL8324383 0.80 ESR1 (0.51) TBXAS1AKR1C3BRS3KDM4EALDH1A1
SCHEMBL14609702 0.75 RECQL (0.51) RECQLAKR1C3KDM4EALDH1A1HPGD
SCHEMBL8322760 0.73 TBXAS1 (0.48) TBXAS1BRS3KDM4EALDH1A1HPGD
SCHEMBL2772402 0.68 TBXAS1 (0.71) RECQLTBXAS1KDM4EALDH1A1SMN1; SMN2
SCHEMBL459101 0.68 TBXAS1 (0.71) RECQLTBXAS1KDM4EALDH1A1SMN1; SMN2
SCHEMBL8322805 0.68 BRS3 (0.48) TBXAS1BRS3KDM4EALDH1A1HPGD
SCHEMBL8322757 0.67 RNASEH1 (0.52) TBXAS1KDM4EALDH1A1SMN1; SMN2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed