SCHEMBL8324544

SCHEMBL8324544

COC(CN)CN(Cc1ccc(F)cc1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.41
YAP1 P46937 1/20 0.39
TEAD4 Q15561 1/20 0.39
TEAD2 Q15562 1/20 0.39
ALDH1A1 P00352 1/20 0.38
PDE6D O43924 1/20 0.38
LMNA P02545 1/20 0.38
ROCK1 Q13464 1/20 0.38
TAS2R14 Q9NYV8 1/20 0.38
RIPK1 Q13546 2/20 0.37
LPAR1 Q92633 2/20 0.37
LPAR5 Q9H1C0 2/20 0.37
NSD2 O96028 1/20 0.36
TSPO P30536 1/20 0.36
POLB P06746 1/20 0.36
APEX1 P27695 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326314 0.87 TDP1 (0.42) TDP1YAP1TEAD4TEAD2ALDH1A1
SCHEMBL8330600 0.85 KDM1A (0.39) YAP1TEAD4TEAD2ROCK1RIPK1
SCHEMBL8328152 0.80 RIPK1 (0.38) TDP1YAP1TEAD4TEAD2ALDH1A1
SCHEMBL7609127 0.75 ALDH1A1 (0.50) TDP1YAP1TEAD4TEAD2ALDH1A1
SCHEMBL8329333 0.73 KDM1A (0.40) TDP1YAP1TEAD4TEAD2RIPK1
SCHEMBL8330238 0.72 TDP1 (0.42) TDP1ALDH1A1LMNATAS2R14RIPK1
SCHEMBL8331046 0.70 CA12 (0.50) TDP1ROCK1POLBAPEX1
SCHEMBL8327663 0.69 ROCK1 (0.44) TDP1YAP1TEAD4TEAD2ALDH1A1
SCHEMBL19545290 0.69 HDAC3 (0.40) YAP1TEAD4TEAD2ROCK1RIPK1
SCHEMBL8328009 0.69 ADRB2 (0.44) TDP1YAP1TEAD4TEAD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed