SCHEMBL8330600

SCHEMBL8330600

COC(CN)CN(Cc1ccc(F)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
KCNQ4 P56696 3/20 0.39
KCNQ5 Q9NR82 3/20 0.39
GRM2 Q14416 1/20 0.38
RIPK1 Q13546 2/20 0.38
NR1D1 P20393 1/20 0.36
BACE1 P56817 3/20 0.36
YAP1 P46937 1/20 0.35
TEAD4 Q15561 1/20 0.35
TEAD2 Q15562 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329333 0.89 KDM1A (0.40) KDM1AHDAC8HDAC6HDAC3HDAC1
SCHEMBL19545290 0.85 HDAC3 (0.40) KDM1AHDAC8HDAC6HDAC3HDAC1
SCHEMBL8324544 0.85 TDP1 (0.41) RIPK1YAP1TEAD4TEAD2ROCK1
SCHEMBL8323152 0.84 KDM1A (0.37) KDM1AHDAC8HDAC6HDAC3HDAC1
SCHEMBL8328376 0.80 CASP3 (0.40) HDAC3HDAC1HDAC2NCOR2BACE1
SCHEMBL2259362 0.80 ROCK1 (0.48) KDM1AHDAC8HDAC6HDAC3HDAC1
SCHEMBL8327226 0.79 HDAC3 (0.41) KDM1AHDAC8HDAC6HDAC3HDAC1
SCHEMBL8331481 0.78 SSTR4 (0.42) KDM1AHDAC8HDAC6HDAC3HDAC1
SCHEMBL8329134 0.78 ROCK1 (0.46) KDM1AHDAC8HDAC6HDAC3HDAC1
SCHEMBL8328955 0.77 HDAC3 (0.43) HDAC8HDAC6HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed