SCHEMBL8324940

SCHEMBL8324940

COC(=O)c1ccc(CCc2cc(Br)ccc2OCc2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 4/20 0.53
ALDH1A1 P00352 2/20 0.52
RAB9A P51151 2/20 0.52
USP28 Q96RU2 1/20 0.52
USP25 Q9UHP3 1/20 0.52
LMNA P02545 5/20 0.51
HTT P42858 2/20 0.51
CCR6 P51684 1/20 0.51
HKDC1 Q2TB90 1/20 0.51
CYP1A2 P05177 3/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
SMPD1 P17405 2/20 0.50
HPGD P15428 2/20 0.50
TP53 P04637 1/20 0.50
ALOX15 P16050 1/20 0.50
ALOX12 P18054 1/20 0.50
CKS1B P61024 1/20 0.50
SKP2 Q13309 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8409537 1.00 CCR5 (0.53) CCR5ALDH1A1RAB9AUSP28USP25
SCHEMBL8318734 0.93 PTGER1 (0.58) CCR5ALDH1A1RAB9AUSP28USP25
SCHEMBL8406894 0.89 HPGD (0.50) ALDH1A1RAB9ALMNACCR6HKDC1
SCHEMBL8408122 0.88 PTGER1 (0.62) CCR5USP28USP25LMNAHTT
SCHEMBL8408175 0.88 HPGD (0.56) ALDH1A1RAB9ALMNACYP1A2CYP3A4
SCHEMBL8406701 0.87 HPGD (0.51) ALDH1A1RAB9ALMNACCR6HKDC1
SCHEMBL8409906 0.86 CCR6 (0.44) CCR5ALDH1A1RAB9AUSP28USP25
SCHEMBL8324992 0.86 CCR5 (0.48) CCR5ALDH1A1RAB9AUSP28USP25
SCHEMBL8406671 0.86 HTR1A (0.66) ALDH1A1RAB9ALMNACYP1A2CYP3A4
SCHEMBL8322935 0.85 CCR5 (0.49) CCR5ALDH1A1RAB9AUSP28USP25

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed
WO-1996011902-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-04-25 WO disclosed